BMS-687453,一种有效的,选择性的PPARα激动剂,对人PPARα的EC50和IC50分别为10 nM和260 nM,较弱地抑制PPARγ的活性,EC50和IC50值分别为4100 nM和>15000 nM
1-(2-Bromoethyl)naphthalene
2-Bromo-3,4-dihydro-6-methoxy-1-[4-(phenylmethoxy)phenyl]naphthalene
1-bromo-2-propoxybenzene
1-[(2-Bromoethyl)sulfanyl]-3-methoxybenzene
1-Bromo-4-cyclobutoxy-benzene
(1S,2R)-2-Fluorocyclopropane-1-carboxylic Acid
Diosbulbin G
Bryonolic acid
23-Oxo-uncaric acid
Methyl 2-(6-acetyl-5-hydroxy-2,3-dihydrobenzofuran-2-yl)propenoate
Erysubin A
Isoastilbin
1-(Pyridin-4-yl)-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one Hydrochloride
1H-Pyrazolo3,4-cpyridin-7-ylamine
2-methyl-2H,6H,7H-pyrazolo[3,4-d]pyridazin-7-one
拉贝地米
顺-2-戊烯-1-醇
3-[(1-hydroxypropan-2-yl)amino]-1λ?-thietane-1,1-dione
6-azaspiro[3,4]octan-7-one
9-methyl-3-oxa-7,9-diazabicyclo[3,3,1]nonanedihydrochloride
2-chloro-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylicacid
2-chloro-7-methoxy-8-methyl-3,4-dihydroquinazolin-4-one
8-bromo-2-chloro-6-fluoroquinazoline
methyl2-{6-chloroimidazo[1,2-b]pyridazin-2-yl}acetate
2-methoxycyclopentan-1-amine
6-methyl-1-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
9-chloro-3,4-dihydro-2H-1,5-benzodioxepine-7-carbaldehyde
N-叔丁基-2-氯吡啶-4-甲酰胺
4-Chloro-6-methoxy[1]benzofuro[3,2-d]pyrimidine
Zimeldine-d6
Rhodamine 800
Mono(2,4-di-tert-butylphenyl)phosphate
5H-indolo[2,1-c][1,4]benzodiazepine-6,12(5aH,7H)-dione
2-t-Butoxypyridine-4-boronic acid pinacol ester
(3-Oxo-thiomorpholin-2-yl)-acetic acid
N'-hydroxy-2-pyrimidinecarboximidamide
4-chloro-2-(4-methoxyphenyl)pyrimidine
替拉曲可
羟乙酸异丙酯
3-溴-2-溴甲基丙酸
3,4-二氯哒嗪
3,4-二硝基氟苯
1-溴-2-萘酚
4-Chloro-7-fluoroindole
6-Methyl-4-nitro indole
5-[(4-ethylphenoxy)methyl]-4-methyl-4H-1,2,4-triazole-3-thiol
4-Ethyl-5-[(4-methylphenoxy)methyl]-4H-1,2,4-triazole-3-thiol
1-(1H-1,2,3-benzotriazole-1-carbothioyl)-1H-1,2,3-benzotriazole
1-(3-氯-4-氟苯基)哌啶
2-[(dimethyl-1H-1,2,4-triazol-1-yl)methyl]piperidine
4,6-二甲基嘧啶
4-吗啉乙酸盐酸盐
4-Hydrazino-6-ethoxyquinoline Hydrochloride
5,8-Dibromo-6-methoxyquinoline
4-chloromethylquinoline hcl
(11β)-11-Hydroxy-17,20:20,21-bis[methylenebis(oxy)]-pregn-5-en-3-one Cyclic 1,2-Ethanediyl Acetal
Helenalin Methacrylate
(S)-(+)-2-氨基丁酰胺盐酸盐
1-氟-2-碘乙烷