AM-4668 是一种GPR40激动剂,用于2 型糖尿病研究。在 A9 细胞中和 CHO 细胞,激活 GPR40 的EC50分别为 3.6 nM 和 36 nM。
| 生物活性 | AM-4668 is aGPR40agonist for type 2 diabetes.EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively[1]. |
| IC50& Target | EC50: 3.6 nM (GPR40, in A9 cells), 36 nM (GPR40, in CHO cells)[1] |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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