Nemonapride 是一种高效的多巴胺 D2受体拮抗剂，其Ki为 0.06 nM。Nemonapride 也能激活5-HT1A受体，其IC50为34 nM。Nemonapride 是一种抗精神病药物，易透过血脑屏障，在动物中表现出强大的抗精神病作用。
| 生物活性 | Nemonapride is a highly potentdopamineD2receptorantagonist with aKiof 0.06 nM. Nemonapride also activates5-HT1Areceptorwith anIC50of 34 nM. Nemonapride is an antipsychotic that readily passes through the blood brain barrier and exhibits potent neuroleptic effects inanimals[1][2][3]. |
| IC50& Target | 5-HT1AReceptor 34 nM (IC50) | D2Receptor 0.06 nM (Ki) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
