DPQ 是一种有效的PARP-1抑制剂。DPQ可降低 N- 甲基 -D- 天冬氨酸 (NMDA) 诱导的 PARP 激活，使 ATP 恢复到接近正常水平，且在 NMDA 严重暴露模型中显著减轻神经元损伤。DPQ 可用于神经保护研究。
| 生物活性 | DPQ is a potentPARP-1inhibitor. DPQ can reduce the N-methyl-d-aspartate (NMDA)-inducedPARPactivation, restoring ATP to near control levels and significantly attenuating neuronal injury in the severe NMDA exposure model. DPQ can be used for researching neuroprotection[1]. |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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