PARP/EZH2-IN-1 是一种PARP(IC506.87 nM)和EZH2(IC5036.51 nM)的双特异性抑制剂,用于治疗野生型BRCA三阴性乳腺癌。
| 生物活性 | PARP/EZH2-IN-1 is a first-in-class dualPARP(IC506.87 nM) andEZH2(IC5036.51 nM) inhibitor for triple-negative breastcancerwith wild-type BRCA. |
| IC50& Target | PARP-1 6.87 nM (IC50) | EZH2 36.51 nM (IC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |