PG106 是一种有效的、选择性的hMC3 receptor拮抗剂 (IC50= 210 nM)，对 hMC4 受体(EC50=9900 nM) 和 hMC5 受体无活性。
| 生物活性 | PG106 is a potent and selectivehuman melanocortin 3 (hMC3) receptorantagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor[1]. |
| IC50& Target | IC50: 210 nM (hMC3 receptor)EC50: 9900 nM (hMC4 receptor)[1] |
| 分子量 | |
| Formula | |
| CAS 号 | |
| Sequence Shortening | Ac-{Nle}-D-{Bal}-{D-Nal}-RWK-NH2 (Lactam bridge:Asp2-Lys7) |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
