SB-277011是可渗透入脑的多巴胺D3受体拮抗剂,对D3,D2,5-HT1D和5-HT1B的pKi分别为8.0,6.0,5.0和<5.2。
| 生物活性 | SB-277011 is a potent and delective dopamine D3 receptor antagonist (pKi values are 8.0, 6.0, 5.0 and<5.2 for D3, D2, 5-HT1D and 5-HT1B respectively); brain penetrant.
IC50 value: 8.0 (pKi)
Target: D3 receptor |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |