Bromodomain inhibitor-10

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CAS NO:

1870849-58-3

Bromodomain inhibitor-10 (compound 128) 是一种有效的溴区结构域bromodomain抑制剂，对 BRD4-1 和 BRD4-2的K_d值分别为 15.0, 2500 nM。Bromodomain inhibitor-10 抑制 IL12p40 的产生。

生物活性

Bromodomain inhibitor-10 (compound 128) is a potentbromodomaininhibitor withK_ds of 15.0, 2500 nM for BRD4-1 and BRD4-2, respectively. Bromodomain inhibitor-10 inhibits the production of IL12p40^[1].

IC₅₀& Target^[1]

BRD4-1

15 nM (Kd)

BRD4-2

2500 nM (Kd)

分子量

364.40

Formula

C₂₀H₂₀N₄O₃

CAS 号

1870849-58-3

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.