OXA(17-33)

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OXA(17-33)

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

343268-91-7

OXA(17-33) 是一种高效、选择性的orexin-1 receptor (OX1)激动剂。OXA(17-33) 对 OX1 (EC₅₀=8.29 nM) 的选择性比 OX2 (187 nM) 高 23 倍。

生物活性

OXA(17-33) is a potent and selectiveorexin-1 receptor (OX1)agonist. OXA(17-33) shows a ~23-fold selectivity for the OX1 (EC₅₀=8.29 nM) over OX2 (187 nM)^[1].

IC₅₀& Target

OX1

8.29 nM (EC₅₀)

OX2

187 nM (EC₅₀)

分子量

1748.98

Formula

C₇₉H₁₂₅N₂₃O₂₂

CAS 号

343268-91-7

Sequence

Tyr-Glu-Leu-Leu-His-Gly-Ala-Gly-Asn-His-Ala-Ala-Gly-Ile-Leu-Thr-Leu-NH2

Sequence Shortening

YELLHGAGNHAAGILTL-NH2

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.