RP101442 是 Ozanimod 的活性代谢物，是一种选择性强的S1PR1激动剂，对 S1PR1 和 S1PR5 的EC50分别为 2.6 nM 和 171 nM。
| 生物活性 | RP101442, an active metabolite of Ozanimod, is a selective, potentS1PR1(sphingosine-1-phosphate receptor 1) agonist, withEC50s of 2.6 nM and 171 nM forS1PR1andS1PR5, respectively[1]. |
| IC50& Target[1] | S1PR1 2.6 nM (EC50) | S1PR5 171 nM (EC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
