AKR1C3-IN-8

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AKR1C3-IN-8

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

AKR1C3-IN-8 (Compound 5) 是一种有效的、选择性的AKR1C3抑制剂，IC₅₀为 0.069 μM。AKR1C3-IN-8 具有抗肿瘤活性。

生物活性	AKR1C3-IN-8 (Compound 5) is a potent, selectiveAKR1C3inhibitor with anIC₅₀of 0.069 μM. AKR1C3-IN-8 shows antitumor activity^[1].
IC₅₀& Target	IC₅₀: 0.069 μM (AKR1C3)^[1]
体外研究 (In Vitro)	AKR1C3-IN-8 (Compound 5) shows antiproliferative activity with an IC₅₀of 52.06 ± 0.99 μM against prostate cancer cell line 22rv1^[1]. AKR1C3-IN-8 (0-50 μM) inhibits PSA expression and testosterone production on 22RV1 cells^[1].
分子量	400.43
Formula	C₂₃H₂₀N₄O₃
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.