Pelubiprofen 是一种具有口服活性,非甾体类抗炎药,是 2-芳基丙酸家族的成员,对COX-2的活性具有相对选择性的作用。Pelubiprofen 抑制 COX 活性和 TGF-β 活化的激酶 1-IκB 激酶 β-NF-κB 途径,并具有显着的抗炎和缓解疼痛作用。
生物活性 | Pelubiprofen, an orally active and non-steroidal anti-inflammatory drug, is a member of the 2-arylpropionic acid family and has relatively selective effects onCOX-2activity. Pelubiprofen inhibitsCOXactivity and thetransforming growth factor-βactivated kinase 1-IκB kinase β-NF-κB pathway, and has significant anti-inflammatory and analgesic effects[1]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |