(R)-Mirtazapine D3 ((R)-Org3770 D3) 是 (R)-Mirtazapine 氘代物。(R)-Mirtazapine 是 Mirtazapine 的 R(–)-对映异构体,在急性热伤害感受动物模型中具有抗伤害感受的作用。(R)-Mirtazapine 是5-HT3受体拮抗剂,在体内主要经 CYP3A4 代谢。
生物活性 | (R)-Mirtazapine D3 ((R)-Org3770 D3) is a deuterium labeled (R)-Mirtazapine. (R)-Mirtazapine is a R(–)-enantiomer of Mirtazapine with antinociceptive properties in an animal model of acute thermal nociception. (R)-Mirtazapine is a5-HT3receptorantagonist. (R)-Mirtazapine is mainly metabolized by CYP3A4[1]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |