Cariprazine D6 (RGH-188 D6) 是 Cariprazine 氘代物。Cariprazine 是一种抗精神病药，结合多巴胺D3,D2和5-HT1A的Ki分别为 0.085 nM，0.49 nM 和 2.6 nM。
| 生物活性 | Cariprazine D6 (RGH-188 D6) is a deuterium labeled Cariprazine. Cariprazine Cariprazine is an antipsychotic agent that exhibits high affinity for theD3(Kiof 0.085 nM) andD2(Kiof 0.49 nM) receptors, and moderate affinity for the5-HT1Areceptor (Kiof 2.6 nM)[1]. |
| IC50& Target | 5-HT1AReceptor 2.6 nM (Ki) | Dopamine D2 Receptor 0.49 nM (Ki) | Dopamine D3 Receptor 0.085 nM (Ki) |
|
| 分子量 | |
| Formula | |
| CAS 号 | |
| 中文名称 | |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
