PARP1-IN-9

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PARP1-IN-9

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

2494000-71-2

PARP1-IN-9 (Compound 5c) 是一种PARP1抑制剂，IC₅₀值为 30.51 nM。PARP1-IN-9 诱导细胞凋亡（apoptosis），具有抗癌活性。PARP1-IN-9 具有高于 Olaparib (HY-10162) 的效果。

生物活性

PARP1-IN-9 (Compound 5c) is aPARP1inhibitor with anIC₅₀of 30.51 nM. PARP1-IN-9 induces cellapoptosisand shows anticancer activity. PARP1-IN-9 has higher potency than Olaparib (HY-10162)^[1].

IC₅₀& Target

PARP1

30.51 nM (IC₅₀)

体外研究
(In Vitro)

PARP1-IN-9 (Compound 5c) shows antiproliferative activity with an IC₅₀of 3.65 μM against MDA-MB-436 cancer cell line^[1].

分子量

359.38

Formula

C₁₈H₂₁N₃O₅

CAS 号

2494000-71-2

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.