PARP1-IN-11 (compound 49) 是一种有效的PARP1抑制剂,其IC50值为 0.082 μM。PARP1-IN-11 显示完全抑制 PARP2 ,并显著抑制 PARP3、TNKS1 和 TNKS2。
| 生物活性 | PARP1-IN-11 (compound 49) is a potentPARP1inhibitor withIC50value of 0.082 μM. PARP1-IN-11 shows complete inhibition ofPARP2and substantially inhibitsPARP3, TNKS1 and TNKS2[1]. |
| IC50& Target[1] | PARP1 0.082 μM (IC50) | PARP2 | TNKS1 | TNKS2 |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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