GSK 4027
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
| CAS: | 2079896-25-4 |
| 分子式: | C17H21BrN4O |
| 分子量: | 377.28 |
| 纯度: | >98% |
| 溶解性: | DMSO : 50 mg/mL (132.53 mM; Need ultrasonic) |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer; Inflammation/Immunology |
| Target: | pIC50: 7.4±0.11 (PCAF) |
| 描述: | GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4±0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. |