(Rac)-NMDARantagonist1是NMDARantagonist1的消旋体。NMDARantagonist1是一种有效且口服生物可利用的，NR2B选择性的NMDAR拮抗剂。
| Cas No. | 2435557-99-4 |
| Canonical SMILES | O=C(NCCC1=CC=C(O)C=C1)C2CCC3=NC4=CC=C(Br)C=C4CN32 |
| 分子式 | C20H20BrN3O2 |
| 分子量 | 414.3 |
| 溶解度 | DMSO: 5 mg/mL (12.07 mM); Water:< 0.1 mg/mL (insoluble) |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | (Rac)-NMDAR antagonist 1 is the racemate of NMDAR antagonist 1. NMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective NMDAR antagonist[1]. [1]. Zhang L, et al. Design, synthesis and bioevaluation of 1,2,3,9-tetrahydropyrrolo[2,1-b]quinazoline-1-carboxylic acid derivatives as potent neuroprotective agents. Eur J Med Chem. 2018 May 10;151:27-38. |
