ATX inhibitor 1是有效的 ATX (IC50=1.23 nM, FS-3; 2.18 nM, bis-pNPP) 抑制剂。
| Cas No. | 2225892-70-4 |
| 分子式 | C21H23Cl2N2O6P |
| 分子量 | 501.3 |
| 溶解度 | DMSO : 250 mg/mL (498.70 mM; Need ultrasonic) |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | ATX inhibitor 1 is a potent ATX (IC50=1.23 nM, FS-3 and 2.18 nM, bis-pNPP) inhibitor. [1]. Balupuri A, et al. Discovery and optimization of ATX inhibitors via modeling, synthesis and biological evaluation. Eur J Med Chem. 2018 Mar 25;148:397-409. |
