SETD2-IN-1 TFA 是一种强效、选择性和口服活性的 SETD2 抑制剂，SETD2 是一种人类组蛋白甲基转移酶。 SETD2-IN-1 TFA 具有抗增殖作用。
| Cas No. | 2411759-92-5 |
| 别名 | SETD2-IN-1 TFA |
| 分子式 | C24H30F4N4O4 |
| 分子量 | 514.51 |
| 溶解度 | DMSO : 200 mg/mL (388.72 mM; Need ultrasonic) |
| 储存条件 | 4°C, away from moisture |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | SETD2-IN-1 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. SETD2-IN-1 TFA has anti-proliferative effects[1]. [1]. John Lampe, et al. Substituted indoles and methods of use thereof. WO2020037079A1. |
