KB-130015 is a novel activator of hERG1 potassium channels, blocking native and recombinant hERG1 channels at high voltages. References: Gessner G, Macianskiene R, Starkus JG, Schonherr R, Heinemann SH. The amiodarone derivative KB130015 activates hERG1 potassium channels via a novel mechanism. Eur J Pharmacol. 2010 Apr 25;632(1-3):52-9. doi: 10.1016/j.ejphar.2010.01.010. PubMed PMID: 20097192; PubMed Central PMCID: PMC2835770.
纯度:≥98%
CAS:147030-48-6