Selective D1-like partial agonist
货号:ajcx26774
CAS:181217-39-0
分子式:C16H16ClNO3.HCl
分子量:342.22
溶解度:Soluble in DMSO
纯度:98%
存储:Store at -20°C
库存:
现货Background:
Selective D1-like dopamine receptor partial agonist (EC50 = 57 nM). Vasodilator in vivo and does not readily cross the blood-brain barrier. Also α2-adrenoceptor antagonist in vitro (Ki = 15 - 25 nM).
Hahn et al (1982) Characterization of the peripheral and central effects of SK&F 82526, a novel DA receptor agonist. J.Pharmacol.Exp.Ther. 223 305 PMID:6127401 |Nichols et al (1990) The pharmacology of fenol. Am.J.Hypertens. 3 116S PMID:1974439 |Sibley et al (1982) Interactions of novel DArgic ligands with D-1 and D-2 DA receptors. Life Sci. 31 637 PMID:6127585