Herkinorin is an analytical reference standard that is functionally categorized as an opioid.
CAS:862073-77-6
分子式:C28H30O8
分子量:494.5
纯度:98%
存储:Store at -20°C
Background:
Herkinorin is an analytical reference standard that is functionally categorized as an opioid. It is a natural neoclerodane diterpene from S. divinorum that preferentially activates the µ-opioid receptor. Unlike the peptide DAMGO , herkinorin activates µ-opioid receptors without inducing arrestin-mediated receptor internalization. Herkinorin has antinociceptive effects in rats. It has been identified as a novel psychoactive substance in multiple agitated emergency department patients screened in a non-targeted manner. This product is intended for research and forensic applications.