生物活性
Tolterodine tartrate (Detrol LA)是毒蕈碱受体拮抗剂。
靶点信息
化学数据
| 目录号 | A10937 |
| 作用机制 | Antagonist (拮抗剂) |
| M. Wt | 475.6 |
| Formula | C26H37NO7 |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles. |
| CAS No. | 124937-52-6 |
| Synonyms | Detrol LA |
| SMILES | CC1=CC(=C(C=C1)O)[C@H](CCN(C(C)C)C(C)C)C2=CC=CC=C2.[C@@H]([C@H](C(=O)O)O)(C(=O)O)O |
溶解度
| In vitro | DMSO | 94 mg/mL (197.66 mM) |
| Water | 17 mg/mL (35.74 mM) |
| Ethanol | 6 mg/mL (12.61 mM) |
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
储备液配制
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
| 0.1 mM | 21.03 mL | 105.13 mL | 210.26 mL |
| 0.5 mM | 4.21 mL | 21.03 mL | 42.05 mL |
| 1 mM | 2.1 mL | 10.51 mL | 21.03 mL |
| 5 mM | 0.42 mL | 2.1 mL | 4.21 mL |
*The above data is based on the productmolecular weight 475.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
