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Pepstatin Ammonium
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
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包装与价格:
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Pepstatin A Ammonium

产品描述

Pepstatin Ammonium is a specific inhibitor of aspartic proteaseproduced by actinomycetes(hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casein-proctase, casein-acid protease and hemoglobin-acid protease with IC50s of 4.5 nM, 6.2 nM, 150 nM, 290 nM, 520 nM and 260 nM , respectively). Pepstatin Ammonium also inhibits HIV protease.

体外活性

Pepstatin inhibits the recombinant HIV protease with an IC50 of 250 μM.

体内活性

Pepstatin suppresses stomach ulceration of the pylorus in ligated Shay rats[1].

Cas No.

T12407

分子式

C34H66N6O9

分子量

702.92

别名

Pepstatin A Ammonium;Pepstatin Ammonium

储存和溶解度

DMSO:41.67 mg/mL (59.28 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
 
 
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