PF4840154 是有效的大鼠和人TrpA1通道选择性激动剂，EC50分别为 97 和 23 nM。PF-4840154 可以诱导 TrpA1 介导的小鼠伤害行为。
产品描述
PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel and elicited TrpA1-mediated nocifensive behaviour in mouse, with EC50 of 97 nM and 23 nM for rTrpA1 and hTrpA1, respectively.
Cas No.
1332708-14-1
分子式
C26H38N6O2
分子量
466.63
储存和溶解度
DMSO:4.66 mg/mL (10 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
