Taltirelin acetate 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM)，能够刺激细胞溶质Ca2+浓度增加 (Ca2+释放) ，其EC50值为 36 nM。
产品描述
Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
Cas No.
1549593-23-8
分子式
C19H27N7O7
分子量
465.46
别名
TA-0910 acetate
储存和溶解度
DMSO:125 mg/mL (268.55 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
