Fasentin 是葡萄糖摄取抑制剂，可抑制GLUT-1/GLUT-4转运蛋白，优先抑制 GLUT4，IC50为 68 μM。它是死亡受体刺激敏化剂，可敏化细胞对 FAS 诱导的细胞死亡，具有抗血管生成活性。
产品描述
Fasentin is an inhibitor of GluT1.
体外活性
Fasentin has been described as a modulator of GLUT-1 and GLUT-4 transporters, thus inhibiting glucose uptake in some cancer cells.
Cas No.
392721-37-8
分子式
C11H9ClF3NO2
分子量
279.64
别名
N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide
储存和溶解度
DMSO:10 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
