Felypressin acetate 是加压素 1 的激动剂，作用于所有精氨酸加压素受体 1AS。 Felypressin acetate 可用于牙科手术。
产品描述
Felypressin acetate is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
体外活性
Felypressin is a synthetic hormone of the posterior pituitary lobe characterized by vasoconstrictor properties mediated by V1 receptors of the blood vessel smooth muscle cells[4].
体内活性
In Wistar rats, Felypressin (240 ng/kg; i.v.) induces a pressor effect and bradycardic effect depending on V1 receptors to induce pressor and bradycardic effects. Felypressin produces a high relationship between bradycardia and mean arterial pressure vari
Cas No.
914453-97-7
分子式
C48H69N13O13S2
分子量
1100.27
别名
PLV 2;PLV-2;醋酸苯赖加压素;PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond);2-(L-Phenylalanine)-8-L-lysinevasopressin
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
