Thermopsoside 是从Aspalathus linearis中分离得到的黄酮衍生物。Thermopsoside 对 CYP450 同工酶有抑制作用,抑制 CYP3A4、CYP2C19、CYP2D6 和 CYP2C9 的IC50的值分别为 6.0 μM、9.5 μM、12.0 μM 和 32.0 μM。
| 生物活性 | Thermopsoside is a flavone derivative isolated fromAspalathus linearis. Thermopsoside exhibits inhibitory effects on CYP450 isozymes withIC50values of 6.0 μM, 9.5 μM, 12.0 μM, 32.0 μM, for CYP3A4, CYP2C19, CYP2D6 and CYP2C9, respectively[1]. |
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| 来源 | - Plants
- Compositae
- Eupatorium japonicumThunb.
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |