BRD0209

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BRD0209

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

1597439-87-6

BRD0209 是一种有效、选择性和双重的GSK3α/β抑制剂 (GSK3αIC₅₀= 19 nM; GSK3βIC₅₀= 5 nM)。BRD0209 还是一种可逆的 ATP 竞争性抑制剂，具有快关动力学 (K_i分别为 4.2 nM)。BRD0209 是一种三环吡唑并四氢喹啉酮化合物。BRD0209 具有研究心境障碍疾病的潜力。

生物活性	BRD0209 is a potent, selective and dual inhibitor ofGSK3α/βinhibitor (GSK3αIC₅₀= 19 nM; GSK3βIC₅₀= 5 nM). BRD0209 is also a reversible ATP-competitive inhibitor with fast-off kinetics (K_i= 4.2 nM, respectively). BRD0209 is a tricyclic pyrazolotetrahydroquinolinone compound. BRD0209 has the potential for the research of mood disorder diseases^[1].
分子量	347.45
Formula	C₂₂H₂₅N₃O
CAS 号	1597439-87-6
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.