BMS-193884 是一种选择性、口服活性和竞争性ETA拮抗剂，对人 ETa受体 (Ki=1.4 nM) 的亲和力是ETB受体的 10000 倍。
| 生物活性 | BMS-193884 is a selective, orally active, and competitiveETAantagonist with 10000-fold greater affinity for the humanETAreceptor (Ki=1.4 nM) than for theETBreceptor[1]. |
| IC50& Target[1] | ETA 1.4 nM (Ki) | ETB 18700 nM (Ki) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
