琥珀酸美托洛尔是一种具有口服活性的选择性 β1-肾上腺素受体拮抗剂。
| Cas No. | 98418-47-4 |
| 别名 | 琥珀酸美托洛尔 |
| 化学名 | 1-(isopropylamino)-3-(4-(2-methoxyethyl)phenoxy)propan-2-ol hemisuccinate |
| Canonical SMILES | OC(COC(C=C1)=CC=C1CCOC)CNC(C)C.OC(COC(C=C2)=CC=C2CCOC)CNC(C)C.OC(CCC(O)=O)=O |
| 分子式 | C34H56N2O10 |
| 分子量 | 652.82 |
| 溶解度 | ≥ 24.75mg/mL in DMSO with gentle warming |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Metoprolol Succinate (Toprol XL) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension.IC50 value:Target: β1 receptor References:
[1]. Benfield P, et al. Metoprolol. An updated review of its pharmacodynamic and pharmacokinetic properties, and therapeutic efficacy, in hypertension, ischaemic heart disease and related cardiovascular disorders. Drugs. 1986 May;31(5):376-429. |
