(E)-8-(3-Chlorostyryl)caffeine 是一种选择性腺苷A2A受体拮抗剂。(E)-8-(3-Chlorostyryl)caffeine 通过独立于其对 A2A受体作用的途径抑制单胺氧化酶 B (MAO-B),Ki值为 70 nM。(E)-8-(3-Chlorostyryl)caffeine 具有用于帕金森病研究的潜力。
生物活性 | (E)-8-(3-Chlorostyryl)caffeine is a selectiveadenosine A2Areceptorantagonist. (E)-8-(3-Chlorostyryl)caffeine inhibitsmonoamine oxidaseB (MAO-B)with aKivalue of 70 nM by a pathway that is independent of its actions on the A2Areceptor. (E)-8-(3-Chlorostyryl)caffeine has the potential for Parkinson's disease research[1]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |